| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | A | | - | Human | 2113 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qim | A | B | n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10661 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5usq | A | B | n-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amine | Human | 7557 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | B | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | 2092 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2j | A | B | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2115 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qik | A | B | n-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10662 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | C | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2104 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2j | A | A | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2124 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | E | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2097 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | A | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | 2095 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | B | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | 2110 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2g | A | B | 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2114 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8u | A | | - | Human | 6616 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5usq | A | A | n-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amine | Human | 7558 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | B | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 6208 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1vjy | A | | 2-[5-(6-methylpyridin-2-yl)-2,3-dihydro-1h-pyrazol-4-yl]-1,5-naphthyridine | Human | 2096 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qil | A | B | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10660 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8s | A | A | - | Human | 6619 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8w | A | A | staurosporine | Human | 6611 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8s | A | B | - | Human | 6609 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e90 | A | B | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6607 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qu0 | A | A | 6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrile | Human | 11967 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | B | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2106 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | E | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2098 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qtz | A | A | 6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridine | Human | 11965 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8t | A | A | - | Human | 6608 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | D | | - | Human | 2126 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e90 | A | A | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6610 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1rw8 | A | | 3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazole | Human | 2100 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5fri | A | B | n-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamide | Human | 6893 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | C | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2093 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 6b8y | A | A | n-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9553 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8z | A | A | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6618 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qu0 | A | B | 6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrile | Human | 11964 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | A | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2127 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qik | A | A | n-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10657 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2k | A | A | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2135 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | C | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2130 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qim | A | A | n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10658 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | D | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2119 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | D | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2132 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2g | A | A | 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2123 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | D | | - | Human | 2131 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | B | | - | Human | 2102 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8x | A | B | staurosporine | Human | 6617 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qil | A | A | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10659 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3gxl | A | | n-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amine | Human | 2116 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | A | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 6207 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qtz | A | B | 6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridine | Human | 11966 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5fri | A | A | n-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamide | Human | 6894 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | D | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2107 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | B | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2121 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2n | A | B | - | Human | 2109 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8z | A | B | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6612 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1py5 | A | | 4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinoline | Human | 2094 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3hmm | A | | 2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amine | Human | 2111 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | C | | - | Human | 2117 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8t | A | B | - | Human | 6613 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | B | | - | Human | 2133 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | A | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2122 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | A | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | 2120 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8x | A | A | staurosporine | Human | 6615 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | F | | - | Human | 2103 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | B | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2108 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wou | A | | 4-({4-[(2,6-dimethylpyridin-3-yl)oxy]pyridin-2-yl}amino)benzenesulfonamide | Human | 2125 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | E | | - | Human | 2134 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2n | A | A | - | Human | 2129 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | A | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2118 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | H | | - | Human | 2099 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 6b8y | A | B | n-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9552 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | E | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2105 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8w | A | B | staurosporine | Human | 6614 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | A | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2112 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | B | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2128 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2k | A | B | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2101 | |