Search results (6 entries covering 4 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
IGF1RInsRTK3d94AB3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amineHuman67600.48
TNK2 (ACK)AckTK4id7Acis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanolHuman34011.00
IGF1RInsRTK8pyiA3-[8-azanyl-1-(4-ethoxy-8-fluoranyl-2-phenyl-quinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutan-1-olHuman149030.43
Btk (BTK)TecTK8fd9AAacalabrutinibMouse148360.40
Btk (BTK)TecTK8fd9ABacalabrutinibMouse148350.40
IGF1RInsRTK3d94AA3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amineHuman67590.48