Search results (10 entries covering 6 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
JAK2JakATK5wevAAn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman83771.00
TGFBR1 (TGFbR1)STKRTKL5friABn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman68930.41
JAK2JakATK4gmyA2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman36840.44
TYK2JakATK4gihAA2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman33390.44
JAK2JakATK5wevABn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman83761.00
TYK2-bJakBTK4oliA2-chloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman21980.41
TYK2JakATK5walABn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman83741.00
TYK2JakATK4gihAB2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman33320.44
TYK2JakATK5walAAn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman83751.00
TGFBR1 (TGFbR1)STKRTKL5friAAn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman68940.41