| KDR | VEGFR | TK | 3c7q | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 5334 | 0.46 | |
| MELK | CAMKL | CAMK | 5maf | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 8732 | 0.46 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | C | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2104 | 0.67 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | E | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2097 | 0.67 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | A | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2127 | 0.67 | |
| GSK3B | GSK | CMGC | 6gjo | A | | (3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-one | Human | 10974 | 0.40 | |
| STK24 (MST3) | STE20 | STE | 4qmt | A | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 5613 | 0.59 | |
| MELK | CAMKL | CAMK | 5mai | A | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8728 | 0.46 | |
| ULK2 | ULK | Other | 6qat | B | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11226 | 1.00 | |
| ULK2 | ULK | Other | 6qat | C | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11232 | 1.00 | |
| RET | Ret | TK | 6nec | A | B | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11150 | 0.46 | |
| ULK2 | ULK | Other | 6qat | D | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11230 | 1.00 | |
| ULK2 | ULK | Other | 6qat | A | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11227 | 1.00 | |
| AAK1 | NAK | Other | 5te0 | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 7156 | 0.46 | |
| MELK | CAMKL | CAMK | 5mai | A | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8730 | 0.46 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6ccf | A | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 9712 | 0.59 | |
| GSK3B | GSK | CMGC | 6gjo | B | | (3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-one | Human | 10973 | 0.40 | |
| RET | Ret | TK | 6nec | C | A | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11147 | 0.46 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6ccf | B | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 9717 | 0.59 | |
| RET | Ret | TK | 6nec | A | A | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11151 | 0.46 | |
| RET | Ret | TK | 6nec | C | B | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11153 | 0.46 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | D | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2107 | 0.67 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | B | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2128 | 0.67 | |
| MAP2K1 | STE7 | STE | 5eym | A | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6969 | 0.46 | |
| MAP2K1 | STE7 | STE | 5eym | B | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6968 | 0.46 | |
| MAP2K1 | STE7 | STE | 5eym | B | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6967 | 0.46 | |
| MAP2K1 | STE7 | STE | 5eym | A | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6966 | 0.46 | |
