| ACVR1 (ALK2) | STKR | TKL | 6szm | A | B | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11737 | 0.72 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | C | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11778 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | D | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1512 | 1.00 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | A | B | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12278 | 0.44 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | A | A | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12277 | 0.44 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | D | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1519 | 1.00 | |
| RIPK2 | RIPK | TKL | 6s1f | D | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11732 | 0.48 | |
| PIM1 | PIM | CAMK | 5toe | A | | 2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrile | Human | 8563 | 0.40 | |
| PIM1 | PIM | CAMK | 5tur | A | | 1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrile | Human | 8565 | 0.41 | |
| RIPK2 | RIPK | TKL | 6s1f | B | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11730 | 0.48 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | A | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1508 | 1.00 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | B | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1514 | 1.00 | |
| RIPK2 | RIPK | TKL | 6s1f | A | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11733 | 0.48 | |
| RIPK2 | RIPK | TKL | 6fu5 | A | | ~{n}-[5-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-phenyl]propane-1-sulfonamide | Human | 9852 | 0.51 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | A | A | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11735 | 0.72 | |
| ACVR1 (ALK2) | STKR | TKL | 8r7g | A | B | 2-fluoranyl-6-methoxy-4-[4-methyl-5-[4-(4-propan-2-ylpiperazin-1-yl)phenyl]pyridin-3-yl]benzamide | Human | 15266 | 0.41 | |
| ACVR1 (ALK2) | STKR | TKL | 8r7g | A | A | 2-fluoranyl-6-methoxy-4-[4-methyl-5-[4-(4-propan-2-ylpiperazin-1-yl)phenyl]pyridin-3-yl]benzamide | Human | 15267 | 0.41 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7z | A | A | 9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridine | Human | 14605 | 0.56 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7z | A | B | 9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridine | Human | 14604 | 0.56 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | B | B | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12275 | 0.44 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | A | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11779 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | D | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11783 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | B | A | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12276 | 0.44 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | B | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1526 | 1.00 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | B | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11781 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | A | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1528 | 1.00 | |
| RIPK2 | RIPK | TKL | 6fu5 | B | | ~{n}-[5-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-phenyl]propane-1-sulfonamide | Human | 9853 | 0.51 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | A | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11784 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | C | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1511 | 1.00 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | B | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11782 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | B | B | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11736 | 0.72 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7w | A | A | 6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepine | Human | 14608 | 0.54 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7w | A | B | 6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepine | Human | 14609 | 0.54 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | C | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11780 | 0.57 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | C | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1522 | 1.00 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | B | A | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11734 | 0.72 | |
| NEK2 | NEK | Other | 2wqo | A | | 4-[2-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]benzoic acid | Human | 331 | 0.41 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | D | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11785 | 0.57 | |
| RIPK2 | RIPK | TKL | 6s1f | C | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11731 | 0.48 | |
