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Search results (14 entries covering 7 PDB structures)
#
Kinase
Family
Group
PDB
Chain
(Alternate) Model
Orthosteric ligand
Organism
Details
Similarity (MFP)
File
PRKAA1 (AMPKa1)
CAMKL
CAMK
7jhg
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
13816
1.00
PRKAA1 (AMPKa1)
CAMKL
CAMK
7m74
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
14017
1.00
ACVR2A (ACTR2)
STKR
TKL
3q4t
B
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2680
1.00
ACVR2A (ACTR2)
STKR
TKL
3q4t
A
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2682
1.00
ACVR1 (ALK2)
STKR
TKL
4c02
A
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
1525
1.00
ACVR2A (ACTR2)
STKR
TKL
3q4t
A
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2686
1.00
ACVR1 (ALK2)
STKR
TKL
3h9r
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
1531
1.00
MELK
CAMKL
CAMK
6gvx
A
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11137
1.00
MELK
CAMKL
CAMK
6gvx
A
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11139
1.00
MELK
CAMKL
CAMK
6gvx
B
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11136
1.00
MELK
CAMKL
CAMK
6gvx
B
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
11138
1.00
ACVR2A (ACTR2)
STKR
TKL
3q4t
B
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
2684
1.00
ACVR1 (ALK2)
STKR
TKL
4c02
A
B
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
1532
1.00
PRKAA2 (AMPKa2)
CAMKL
CAMK
3aqv
A
6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
Human
193
1.00
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